Best Peptides for Weight Loss

Weight loss peptides — particularly GLP-1 receptor agonists like Semaglutide and Tirzepatide — have become the most commercially significant peptide class in recent years. These compounds work by mimicking incretin hormones that regulate appetite, blood sugar, and metabolic rate.

The metabolic peptides listed below range from FDA-approved medications to experimental research compounds. We present the evidence objectively: what the clinical trials actually show, what the dosing protocols look like, and what side effects have been documented.

Peptides for Weight Loss Peptides

  • 5-Amino-1MQ — 5-Amino-1MQ is a small molecule inhibitor of nicotinamide N-methyltransferase (NNMT), an enzyme linked to obesity and...
  • AOD-9604 — AOD-9604 is a modified C-terminal fragment of human growth hormone (amino acids 176-191). Originally developed as an...
  • HGH Fragment 176-191 — HGH Fragment 176-191 is a stabilized fragment of the C-terminal portion of human growth hormone (amino acids 176-191)....
  • Liraglutide — Liraglutide is a GLP-1 receptor agonist with 97% sequence homology to native GLP-1. FDA-approved as Victoza (diabetes)...
  • Retatrutide — Retatrutide is an investigational triple agonist targeting GIP, GLP-1, and glucagon receptors simultaneously. Phase 2...
  • Semaglutide — Semaglutide is a GLP-1 receptor agonist with 94% sequence homology to human glucagon-like peptide-1. Used for weight...
  • Tirzepatide — Tirzepatide is a dual GIP/GLP-1 receptor agonist for weight management and type 2 diabetes. Marketed as Mounjaro...

Frequently Asked Questions

What is the most effective weight loss peptide?

Based on clinical trial data, Tirzepatide (a dual GIP/GLP-1 agonist) has shown the largest average weight loss in Phase 3 trials — up to 22.5% body weight reduction at the highest dose. Semaglutide 2.4mg (Wegovy) showed approximately 15% average weight loss. Retatrutide (a triple agonist) showed up to 24% in Phase 2 trials.

Are weight loss peptides FDA approved?

Semaglutide (as Wegovy/Ozempic) and Tirzepatide (as Mounjaro/Zepbound) are FDA-approved for weight management or type 2 diabetes. Other metabolic peptides like AOD-9604, Retatrutide, and 5-Amino-1MQ are not FDA-approved and remain in research stages.

How do GLP-1 peptides cause weight loss?

GLP-1 receptor agonists reduce appetite by acting on brain regions that control hunger and satiety, slow gastric emptying (making you feel full longer), and improve insulin sensitivity. Dual and triple agonists like Tirzepatide and Retatrutide add GIP and/or glucagon receptor activation for additional metabolic effects.

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