PE-22-28

PE-22-28 is a synthetic 7-amino-acid peptide derived from the spadin family, designed to inhibit the TREK-1 potassium channel. Research focuses on antidepressant-like effects and cognitive enhancement through BDNF-mediated neuroplasticity in preclinical models.

At a Glance

Summary: Inhibits TREK-1 potassium channels to enhance serotonergic neurotransmission and rapidly upregulate BDNF, producing antidepressant and cognitive-enhancing effects. Mechanisms (reported/proposed across domains): Mood / antidepressant • Blocks TREK-1 (TWIK-Related K+ Channel 1), a background potassium channel whose deletion in mice produces a depression-resistant phenotype. • TREK-1...

Safety Profile

Investigational - Preclinical Only

Research Dosing

Dose: 100–500 mcg (estimated from preclinical data) · Route: Intranasal · Subcutaneous (SC) · Frequency: 1× daily · Duration: 2–4 weeks

Categories

  • Research Only
  • Cognitive Function
  • Nootropic
  • BDNF Enhancement
  • Stress Reduction
  • Preclinical Evidence
  • Not FDA Approved
  • Intranasal Available

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